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5JWM

3D Structure View

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GENERAL
TITLE
BIVALENT BET BROMODOMAIN INHIBITION
DATE LAST MODIFIED
Sep 27, 2023
RELEASE
Jul 6, 2016
CLASSIFICATION
TRANSCRIPTION/TRANSCRIPTION INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 2 2 21
RESOLUTION RANGE HIGH
1.71
RESOLUTION RANGE LOW
43.56
PUBMED ID
DOI
10.1038/NCHEMBIO.2209
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
O60885 BRD4, HUNK1 ESCHERICHIA COLI HUMAN
PROTEIN HUNK1
Mutations
O60885 BRD4, HUNK1 ESCHERICHIA COLI HUMAN
PROTEIN HUNK1
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402